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Alan D. Borthwick · Study
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Author
Alan D. Borthwick
4 works
· latest 2012
· 1 institutions
cluster: provisional
ORCID 0000-0002-6740-4232
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Citations
300
Works here
4
05
07
12
Most cited in this library
The discovery of GSK221149A: A potent and selective oxytocin antagonist
2007 · 91 citations
Pyridyl-2,5-Diketopiperazines as Potent, Selective, and Orally Bioavailable Oxytocin Antagonists: Synthesis, Pharmacokinetics, and In Vivo Potency
2012 · 89 citations
2,5-Diketopiperazines as potent and selective oxytocin antagonists 1: identification, stereochemistry and initial SAR
2005 · 67 citations
2,5-Diketopiperazines as Potent, Selective, and Orally Bioavailable Oxytocin Antagonists. 2. Synthesis, Chirality, and Pharmacokinetics
2005 · 53 citations
Works
4 shown
Pyridyl-2,5-Diketopiperazines as Potent, Selective, and Orally Bioavailable Oxytocin Antagonists: Synthesis, Pharmacokinetics, and In Vivo Potency
Journal of Medicinal Chemistry
·
2012
·
16 authors
89
citations
The discovery of GSK221149A: A potent and selective oxytocin antagonist
Bioorganic & Medicinal Chemistry Letters
·
2007
·
22 authors
91
citations
2,5-Diketopiperazines as Potent, Selective, and Orally Bioavailable Oxytocin Antagonists. 2. Synthesis, Chirality, and Pharmacokinetics
Journal of Medicinal Chemistry
·
2005
·
11 authors
53
citations
2,5-Diketopiperazines as potent and selective oxytocin antagonists 1: identification, stereochemistry and initial SAR
Bioorganic & Medicinal Chemistry Letters
·
2005
·
12 authors
67
citations